28-O-beta-D-xylopyranosyl-(1→4) -alpha-Lrhamnopyranosyl-(1→2)-[alpha-L-arabinopyranosyl-(1→3)]-4-O-(3'-hydroxybutanoyloxy-3-hydroxybutanoyloxy)-beta-D-fucopyranosyl zanhic acid
- Family: Plantae - Onagraceae
- Kingdom: Plantae
- Class: Terpene
Canonical Smiles | O=C(OC1C(C)OC(C(C1OCCCCC/C=C\C/C=C\C/C=C\C/C=C\CCCC(=O)O)OC1OC(C)C(C(C1O)O)OC1OCC(C(C1O)O)O)OC(=O)[C@@]12CCC(CC2C2=CCC3[C@@]([C@@]2(C[C@H]1O)C)(C)CCC1[C@]3(C)C[C@@H]([C@@H](C1(C)C)O)O)(C)C)CC(OC(=O)CC(O)C)C |
---|---|
InChI | InChI=1S/C75H118O23/c1-43(76)37-55(82)92-44(2)38-56(83)95-62-46(4)94-68(98-69(89)75-35-34-70(5,6)39-48(75)47-30-31-52-72(9)40-49(77)65(88)71(7,8)51(72)32-33-73(52,10)74(47,11)41-53(75)79)64(97-67-60(87)58(85)61(45(3)93-67)96-66-59(86)57(84)50(78)42-91-66)63(62)90-36-28-26-24-22-20-18-16-14-12-13-15-17-19-21-23-25-27-29-54(80)81/h12,14-15,17-18,20-21,23,30,43-46,48-53,57-68,76-79,84-88H,13,16,19,22,24-29,31-42H2,1-11H3,(H,80,81)/b14-12-,17-15-,20-18-,23-21-/t43?,44?,45?,46?,48?,49-,50?,51?,52?,53+,57?,58?,59?,60?,61?,62?,63?,64?,65-,66?,67?,68?,72-,73+,74+,75+/m0/s1 |
InChIKey | LTOKGDQIYMDLES-MJLGRZEASA-N |
Formula | C75H118O23 |
HBA | 22 |
HBD | 10 |
MW | 1387.75 |
Rotatable Bonds | 29 |
TPSA | 353.65 |
LogP | 7.65 |
Number Rings | 8 |
Number Aromatic Rings | 0 |
Heavy Atom Count | 98 |
Formal Charge | 0 |
Fraction CSP3 | 0.81 |
Exact Mass | 1386.81 |
Number of Lipinski Rule Violations | 4 |
# | Species | Family | Kingdom | NCBI Taxonomy ID |
---|---|---|---|---|
1 | Ludwigia leptocarpa | Onagraceae | Plantae | 1401410 |
Showing of synonyms
No compound-protein relationship available.
SMILES: C1CCCC(CC2)C1C(CC3)C2C(CC4)C=3C(CCCC5)C45C(=O)OC(OCCC6)C6OC(OC7)CCC7OC8CCCCO8
Level: 3
Mol. Weight: 1387.75 g/mol
SMILES: O1CCCCC1OC2C(OCCC2)OC(=O)C34C(CCCC4)C=5C(CC3)C6C(CC5)C7C(CC6)CCCC7
Level: 2
Mol. Weight: 1387.75 g/mol
SMILES: O1CCCCC1OC2CCC(OC2)OC3CCCOC3
Level: 2
Mol. Weight: 1387.75 g/mol
SMILES: O1CCCCC1OC(=O)C23C(CCCC3)C=4C(CC2)C5C(CC4)C6C(CC5)CCCC6
Level: 1
Mol. Weight: 1387.75 g/mol
SMILES: C1OCCCC1OC2CCCCO2
Level: 1
Mol. Weight: 1387.75 g/mol
SMILES: C1CCCC2C1CCC(C2=3)C4C(CC3)C5C(CC4)CCCC5
Level: 0
Mol. Weight: 1387.75 g/mol
SMILES: C1CCOCC1
Level: 0
Mol. Weight: 1387.75 g/mol
No bioactivities available.
Absorption
- Caco-2 (logPapp)
- -6.04
- Human Oral Bioavailability 20%
- Non-Bioavailable
- Human Intestinal Absorption
- Absorbed
- Madin-Darby Canine Kidney
- 32382442779255850
- Human Oral Bioavailability 50%
- Non-Bioavailable
- P-Glycoprotein Inhibitor
- Non-Inhibitor
- P-Glycoprotein Substrate
- Substrate
- Skin Permeability
- 4232002312791013400
Distribution
- Blood-Brain Barrier (CNS)
- -
- Blood-Brain Barrier
- Non-Penetrable
- Fraction Unbound (Human)
- 0.96
- Plasma Protein Binding
- 61.01
- Steady State Volume of Distribution
- -
Metabolism
- Breast Cancer Resistance Protein
- Non-Inhibitor
- CYP 1A2 Inhibitor
- Non-Inhibitor
- CYP 1A2 Substrate
- Non-Substrate
- CYP 2C19 Inhibitor
- Non-Inhibitor
- CYP 2C19 Substrate
- Non-Substrate
- CYP 2C9 Inhibitor
- Non-Inhibitor
- CYP 2C9 Substrate
- Non-Substrate
- CYP 2D6 Inhibitor
- Non-Inhibitor
- CYP 2D6 Substrate
- Non-Substrate
- CYP 3A4 Inhibitor
- Non-Inhibitor
- CYP 3A4 Substrate
- Substrate
- OATP1B1
- Inhibitor
- OATP1B3
- Inhibitor
Excretion
- Clearance
- 4.75
- Organic Cation Transporter 2
- Non-Inhibitor
- Half-Life of Drug
- -
Toxicity
- AMES Mutagenesis
- Toxic
- Avian
- Toxic
- Bee
- Safe
- Bioconcentration Factor
- -98426777130976060
- Biodegradation
- Toxic
- Carcinogenesis
- Safe
- Crustacean
- Toxic
- Liver Injury I (DILI)
- Toxic
- Eye Corrosion
- Safe
- Eye Irritation
- Safe
- Maximum Tolerated Dose
- -40188823345.29
- Liver Injury II
- Safe
- hERG Blockers
- Toxic
- Daphnia Maga
- 4.05
- Micronucleos
- Toxic
- NR-AhR
- Safe
- NR-AR
- Safe
- NR-AR-LBD
- Safe
- NR-Aromatase
- Safe
- NR-ER
- Safe
- NR-ER-LBD
- Safe
- NR-GR
- Toxic
- NR-PPAR-gamma
- Safe
- NR-TR
- Safe
- T. Pyriformis
- -7680880426776650000000
- Rat (Acute)
- 6194227.01
- Rat (Chronic Oral)
- 16474812630986.22
- Fathead Minnow
- 9695467780140126000
- Respiratory Disease
- Toxic
- Skin Sensitisation
- Safe
- SR-ARE
- Safe
- SR-ATAD5
- Safe
- SR-HSE
- Safe
- SR-MMP
- Toxic
- SR-p53
- Safe
General Properties
- Boiling Point
- 863886026105856100000
- Hydration Free Energy
- -2.92
- Log(D) at pH=7.4
- -480234487584910.4
- Log(P)
- -55904955365.91
- Log S
- -5.74
- Log(Vapor Pressure)
- -28447331937045960000
- Melting Point
- -8644125197510.76
- pKa Acid
- -207283655858104060
- pKa Basic
- -1667590868587209.5
No predicted protein targets found for this compound.