Vaccaroside D
- Family: Plantae - Caryophyllaceae
- Kingdom: Plantae
-
Class: Saponin
- Subclass: Triterpene Saponin
Canonical Smiles | OCCC[C@@]1(C)[C@@H](CC[C@@]2([C@@H]1CC=C1[C@@]2(C)CC[C@@]2([C@H]1CC(C)(C)CC2)C(=O)O[C@@H]1O[C@H](CO[C@@H]2O[C@H](CO)[C@H]([C@@H]([C@H]2O[C@@H]2O[C@H](CO)[C@H]([C@@H]([C@H]2O)O)O)O)O)[C@H]([C@@H]([C@H]1O)O[C@@H]1O[C@H](CO)[C@H]([C@@H]([C@H]1O)O)O)O)C)C(=C)C(=O)O |
---|---|
InChI | InChI=1S/C54H86O25/c1-23(44(69)70)24-10-12-53(6)31(51(24,4)11-7-17-55)9-8-25-26-18-50(2,3)13-15-54(26,16-14-52(25,53)5)49(71)79-47-41(68)42(77-45-39(66)36(63)32(59)27(19-56)73-45)35(62)30(76-47)22-72-48-43(38(65)34(61)29(21-58)75-48)78-46-40(67)37(64)33(60)28(20-57)74-46/h8,24,26-43,45-48,55-68H,1,7,9-22H2,2-6H3,(H,69,70)/t24-,26-,27+,28+,29+,30+,31+,32+,33+,34+,35+,36-,37-,38-,39+,40+,41+,42-,43+,45-,46-,47-,48+,51-,52+,53+,54-/m0/s1 |
InChIKey | QCSJRNNSTFHPAZ-SNDIJUFTSA-N |
Formula | C54H86O25 |
HBA | 24 |
HBD | 15 |
MW | 1135.26 |
Rotatable Bonds | 17 |
TPSA | 411.43 |
LogP | -2.8 |
Number Rings | 8 |
Number Aromatic Rings | 0 |
Heavy Atom Count | 79 |
Formal Charge | 0 |
Fraction CSP3 | 0.89 |
Exact Mass | 1134.55 |
Number of Lipinski Rule Violations | 3 |
# | Species | Family | Kingdom | NCBI Taxonomy ID |
---|---|---|---|---|
1 | Vaccaria pyramidata | Caryophyllaceae | Plantae | 39387 |
Showing of synonyms
- Said R, Hamed A, et al. (2019). Flavone C-glycosides from Vaccaria pyramidata: Structure elucidation by spectroscopy and theoretical calculations. Phytochemistry Letters, 2019, 29, 119-124. [View]
No compound-protein relationship available.
SMILES: C1CCCC(CC2)C1C(CC3)C=2C(CCCC4)C34C(=O)OC(O5)CC(OC6CCCCO6)CC5COC(OCCC7)C7OC8CCCCO8
Level: 4
Mol. Weight: 1135.26 g/mol
SMILES: C1CCCC(CC2)C1C(CC3)C=2C(CCCC4)C34C(=O)OC(O5)CCCC5COC(OCCC6)C6OC7CCCCO7
Level: 3
Mol. Weight: 1135.26 g/mol
SMILES: C1CCCC(CC2)C1C(CC3)C=2C(CCCC4)C34C(=O)OC(O5)CC(OC6CCCCO6)CC5COC7CCCCO7
Level: 3
Mol. Weight: 1135.26 g/mol
SMILES: O1CCCCC1OC(CCO2)CC2COC(OCCC3)C3OC4CCCCO4
Level: 3
Mol. Weight: 1135.26 g/mol
SMILES: C1CCCC(CC2)C1C(CC3)C=2C(CCCC4)C34C(=O)OC(O5)CCCC5COC6CCCCO6
Level: 2
Mol. Weight: 1135.26 g/mol
SMILES: C1CCCC(CC2)C1C(CC3)C=2C(CCCC4)C34C(=O)OC(OCC5)CC5OC6CCCCO6
Level: 2
Mol. Weight: 1135.26 g/mol
SMILES: O1CCCCC1OCC2CC(CCO2)OC3CCCCO3
Level: 2
Mol. Weight: 1135.26 g/mol
SMILES: O1CCCCC1COC(OCCC2)C2OC3CCCCO3
Level: 2
Mol. Weight: 1135.26 g/mol
SMILES: O1CCCCC1OC(=O)C23C(CCCC3)C=4C(CC2)C5C(CC4)CCCC5
Level: 1
Mol. Weight: 1135.26 g/mol
SMILES: O1CCCCC1COC2CCCCO2
Level: 1
Mol. Weight: 1135.26 g/mol
SMILES: C1OCCCC1OC2CCCCO2
Level: 1
Mol. Weight: 1135.26 g/mol
SMILES: C1COCCC1OC2CCCCO2
Level: 1
Mol. Weight: 1135.26 g/mol
SMILES: C1CCCC(CC2)C1C(C=23)CCC4C3CCCC4
Level: 0
Mol. Weight: 1135.26 g/mol
SMILES: C1CCOCC1
Level: 0
Mol. Weight: 1135.26 g/mol
No bioactivities available.
Absorption
- Caco-2 (logPapp)
- -6.42
- Human Oral Bioavailability 20%
- Non-Bioavailable
- Human Intestinal Absorption
- Non-Absorbed
- Madin-Darby Canine Kidney
- 2065687.11
- Human Oral Bioavailability 50%
- Non-Bioavailable
- P-Glycoprotein Inhibitor
- Non-Inhibitor
- P-Glycoprotein Substrate
- Non-Substrate
- Skin Permeability
- 269962065.43
Distribution
- Blood-Brain Barrier (CNS)
- -
- Blood-Brain Barrier
- Non-Penetrable
- Fraction Unbound (Human)
- 0.79
- Plasma Protein Binding
- 62.86
- Steady State Volume of Distribution
- -
Metabolism
- Breast Cancer Resistance Protein
- Non-Inhibitor
- CYP 1A2 Inhibitor
- Non-Inhibitor
- CYP 1A2 Substrate
- Non-Substrate
- CYP 2C19 Inhibitor
- Non-Inhibitor
- CYP 2C19 Substrate
- Non-Substrate
- CYP 2C9 Inhibitor
- Non-Inhibitor
- CYP 2C9 Substrate
- Non-Substrate
- CYP 2D6 Inhibitor
- Non-Inhibitor
- CYP 2D6 Substrate
- Non-Substrate
- CYP 3A4 Inhibitor
- Non-Inhibitor
- CYP 3A4 Substrate
- Substrate
- OATP1B1
- Inhibitor
- OATP1B3
- Non-Inhibitor
Excretion
- Clearance
- 1.21
- Organic Cation Transporter 2
- Non-Inhibitor
- Half-Life of Drug
- -
Toxicity
- AMES Mutagenesis
- Safe
- Avian
- Toxic
- Bee
- Safe
- Bioconcentration Factor
- -6278695.42
- Biodegradation
- Toxic
- Carcinogenesis
- Safe
- Crustacean
- Toxic
- Liver Injury I (DILI)
- Toxic
- Eye Corrosion
- Safe
- Eye Irritation
- Safe
- Maximum Tolerated Dose
- -3.34
- Liver Injury II
- Safe
- hERG Blockers
- Toxic
- Daphnia Maga
- 4.05
- Micronucleos
- Toxic
- NR-AhR
- Safe
- NR-AR
- Safe
- NR-AR-LBD
- Safe
- NR-Aromatase
- Safe
- NR-ER
- Safe
- NR-ER-LBD
- Safe
- NR-GR
- Safe
- NR-PPAR-gamma
- Safe
- NR-TR
- Safe
- T. Pyriformis
- -489968116774.07
- Rat (Acute)
- 3.51
- Rat (Chronic Oral)
- 1050.41
- Fathead Minnow
- 618480513.88
- Respiratory Disease
- Toxic
- Skin Sensitisation
- Safe
- SR-ARE
- Safe
- SR-ATAD5
- Safe
- SR-HSE
- Safe
- SR-MMP
- Safe
- SR-p53
- Safe
General Properties
- Boiling Point
- 55107829341.13
- Hydration Free Energy
- -2.92
- Log(D) at pH=7.4
- -30626.74
- Log(P)
- -3.4
- Log S
- -2.39
- Log(Vapor Pressure)
- -1814672826.28
- Melting Point
- 126.3
- pKa Acid
- -13222658.29
- pKa Basic
- -106364.81
No predicted protein targets found for this compound.