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263 Families
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| # | Family | Kingdom | #Compounds | #Species |
| 1 | Acanthaceae | Plantae | 79 | 12 |
| 2 | Achariaceae | Plantae | 10 | 1 |
| 3 | Actiinidae | Animalia | 1 | 1 |
| 4 | Adoxaceae | Plantae | 12 | 1 |
| 5 | Agaricaceae | Fungi | 5 | 1 |
| 6 | Agavaceae | Plantae | 42 | 6 |
| 7 | Aizoaceae | Plantae | 6 | 1 |
| 8 | Alcyoniidae | Animalia | 93 | 11 |
| 9 | Alysseae | Plantae | 5 | 1 |
| 10 | Amaranthaceae | Plantae | 40 | 7 |
| 11 | Amaryllidaceae | Plantae | 120 | 19 |
| 12 | Amphisphaeriaceae | Fungi | 10 | 1 |
| 13 | Anacardiaceae | Plantae | 139 | 21 |
| 14 | Anchinoidae | Animalia | 3 | 2 |
| 15 | Ancistrocladaceae | Plantae | 150 | 10 |
| 16 | Annonaceae | Plantae | 283 | 39 |
| 17 | Apiaceae | Plantae | 389 | 37 |
| 18 | Apidae | Animalia | 67 | 3 |
| 19 | Aplysiidae | Animalia | 2 | 1 |
| 20 | Aplysinellidae | Animalia | 15 | 1 |
| 21 | Apocynaceae | Plantae | 351 | 39 |
| 22 | Arabideae | Plantae | 6 | 1 |
| 23 | Araceae | Plantae | 2 | 1 |
| 24 | Araliaceae | Plantae | 109 | 10 |
| 25 | Araucariaceae | Plantae | 10 | 1 |
| 26 | Archaeidae | Animalia | 2 | 1 |
| 27 | Arecaceae | Plantae | 104 | 12 |
| 28 | Aristolochiaceae | Plantae | 3 | 2 |
| 29 | Ascidiaceae | Animalia | 2 | 1 |
| 30 | Asclepiadaceae | Plantae | 5 | 3 |
| 31 | Asparagaceae | Plantae | 44 | 6 |
| 32 | Asphodelaceae | Plantae | 195 | 43 |
| 33 | Asteraceae-Compositae | Plantae | 1765 | 264 |
| 34 | Avicenniaceae | Plantae | 5 | 1 |
| 35 | Axinellidae | Animalia | 4 | 1 |
| 36 | Azzolaceae | Plantae | 9 | 1 |
| 37 | Bacillaceae | Monera | 1 | 1 |
| 38 | Berberidaceae | Plantae | 2 | 2 |
| 39 | Bignoniaceae | Plantae | 109 | 15 |
| 40 | Bionectriaceae | Fungi | 10 | 1 |
| 41 | Bombacaceae | Plantae | 14 | 2 |
| 42 | Boraginaceae | Plantae | 116 | 18 |
| 43 | Botryosphaeriaceae | Fungi | 21 | 2 |
| 44 | Bovidae | Animalia | 36 | 3 |
| 45 | Brassicaceae | Plantae | 67 | 11 |
| 46 | Burseraceae | Plantae | 224 | 11 |
| 47 | Cactaceae | Plantae | 7 | 2 |
| 48 | Caesalpiniaceae | Plantae | 15 | 3 |
| 49 | Caesalpinioideae | Plantae | 14 | 1 |
| 50 | Callyspongiidae | Animalia | 43 | 6 |
| 51 | Calophyllaceae | Plantae | 2 | 1 |
| 52 | Campanulaceae | Plantae | 14 | 2 |
| 53 | Canellaceae | Plantae | 39 | 2 |
| 54 | Cannabaceae | Plantae | 29 | 1 |
| 55 | Capparaceae | Plantae | 155 | 14 |
| 56 | Caprifoliaceae | Plantae | 30 | 2 |
| 57 | Caryophyllaceae | Plantae | 84 | 15 |
| 58 | Cecropiaceae | Plantae | 11 | 1 |
| 59 | Celastraceae | Plantae | 55 | 5 |
| 60 | Chaetomiaceae | Fungi | 44 | 16 |
| 61 | Chaetosphaeriales | Fungi | 2 | 1 |
| 62 | Chenopodiaceae | Plantae | 188 | 16 |
| 63 | Chromodorididae | Animalia | 7 | 1 |
| 64 | Chrysobalanaceae | Plantae | 6 | 1 |
| 65 | Cistaceae | Plantae | 57 | 5 |
| 66 | Clavelinidae | Animalia | 3 | 2 |
| 67 | Cleomaceae | Plantae | 6 | 1 |
| 68 | Clusiaceae | Plantae | 70 | 10 |
| 69 | Clusiaceae-Guttiferae | Plantae | 9 | 2 |
| 70 | Combretaceae | Plantae | 87 | 14 |
| 71 | Commelinaceae | Plantae | 9 | 1 |
| 72 | Convolvulaceae | Plantae | 38 | 7 |
| 73 | Corallinaceae | Plantae | 7 | 1 |
| 74 | Cordycipitaceae | Fungi | 11 | 2 |
| 75 | Cruciferae | Plantae | 4 | 1 |
| 76 | Cruciferae-Brassicaceea | Plantae | 76 | 5 |
| 77 | Cucurbitaceae | Plantae | 43 | 6 |
| 78 | Cupressaceae | Plantae | 225 | 10 |
| 79 | Cyperaceae | Plantae | 34 | 5 |
| 80 | Cypress | Fungi | 9 | 1 |
| 81 | Cystoseiraceae | Plantae | 3 | 2 |
| 82 | Dematiaceae | Fungi | 8 | 1 |
| 83 | Dendrophylliidae | Animalia | 10 | 1 |
| 84 | Desmacellidae | Animalia | 8 | 1 |
| 85 | Diadematidae | Plantae | 4 | 1 |
| 86 | Dichapetalaceae | Plantae | 4 | 1 |
| 87 | Dictyonellidae | Animalia | 12 | 1 |
| 88 | Dictyotaceae | Plantae | 12 | 4 |
| 89 | Didemnidae | Animalia | 2 | 1 |
| 90 | Didymellaceae | Fungi | 9 | 1 |
| 91 | Dilleniaceae | Plantae | 4 | 1 |
| 92 | Dioncophyllaceae | Plantae | 14 | 2 |
| 93 | Dioscoreaceae | Plantae | 20 | 3 |
| 94 | Dipsacaceae | Plantae | 5 | 2 |
| 95 | Dipterocarpaceae | Plantae | 23 | 1 |
| 96 | Dracaenaceae | Plantae | 51 | 3 |
| 97 | Dysideidae | Animalia | 2 | 1 |
| 98 | Ebenaceae | Plantae | 34 | 6 |
| 99 | Ephedraceae | Plantae | 16 | 2 |
| 100 | Equisetaceae | Plantae | 2 | 1 |